Design, synthesis and evaluation of novel activity-based probes and inhibitors for trypsin-like serine proteases : focus on Dry eye disease (DED) and Irritable bowel syndrome (IBS)

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Antwerp, University of Antwerp, Faculty of Pharmaceutical, Biomedical and Veterinary Sciences, Department of Pharmaceutical Sciences, 2023,xi, 289

Chemically diverse activity-based probes with unexpected inhibitory mechanisms targeting trypsin-like serine proteases

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Frontiers in Chemistry - ISSN 2296-2646-10 (2023) p. 1-17
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Improved synthesis of the selected serine protease uPA inhibitor UAMC-00050, a lead compound for the treatment of dry eye disease

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Organic process research and development - ISSN 1083-6160-26:10 (2022) p. 2937-2946
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